Title of article
Facile preparation of N-acylsulfonamides by using sulfonyl isocyanate
Author/Authors
Manabe، نويسنده , , Shino and Sugioka، نويسنده , , Tomoyuki and Ito، نويسنده , , Yukishige، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2007
Pages
3
From page
787
To page
789
Abstract
N-Acylsulfonamide is widely used as a carboxylic acid bioisostere. A rapid and mild acyl sulfonamide preparation methodology from carboxylic acid and arylsulfonyl isocyanate in the presence of amine is described. The preparation of biologically active acylsulfonamide by our methodology is also presented.
Keywords
N-Acylsulfonamide , Sulfonyl isocyanate , Carboxylic acid isostere
Journal title
Tetrahedron Letters
Serial Year
2007
Journal title
Tetrahedron Letters
Record number
1854070
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