Title of article
Selective palladium-catalyzed amination of the heterocyclic core of variolins
Author/Authors
Baeza، نويسنده , , Alejandro and Burgos، نويسنده , , Carolina and Alvarez-Builla، نويسنده , , Julio and Vaquero، نويسنده , , Juan J.، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2007
Pages
5
From page
2597
To page
2601
Abstract
A new and selective palladium-catalyzed amination of the pyrido[3′,3′:4,5]pyrrolo[1,2-c]pyrimidine nucleus, the heterocyclic core of the variolin alkaloids, is described. The method allows the introduction of amino and aryl- and alkylamino substituents on the C9 position in advanced precursors of variolin B and deoxyvariolin.
Keywords
3?:4 , 2-c]pyrimidine , N-Tosylmethyl dichloroformimide , Palladium-catalyzed , amination , Variolins
Journal title
Tetrahedron Letters
Serial Year
2007
Journal title
Tetrahedron Letters
Record number
1854683
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