Title of article
Development of copper-mediated allylation of γ-activated-α,β-unsaturated lactam toward peptide mimetic synthesis
Author/Authors
Sasaki، نويسنده , , Yoshikazu and Yamaguchi، نويسنده , , Keiko and Tsuji، نويسنده , , Takashi and Shigenaga، نويسنده , , Akira and Fujii، نويسنده , , Nobutaka and Otaka، نويسنده , , Akira، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2007
Pages
4
From page
3221
To page
3224
Abstract
Reactions of γ-activated-α,β-unsaturated lactams with allylboronate in the presence of LiOi-Pr and CuX (stoichiometric or catalytic amount) proceed in an anti-SN2′ manner to yield α-allylated compounds that serve as a potential synthetic intermediate for cis-aminoacyl-Pro mimetics.
Keywords
proline , Copper-mediated anti-SN2? , Dipeptide mimetic , allylation
Journal title
Tetrahedron Letters
Serial Year
2007
Journal title
Tetrahedron Letters
Record number
1854878
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