• Title of article

    Pot, atom and step economic (PASE) synthesis of highly functionalized piperidines: a five-component condensation

  • Author/Authors

    Clarke، نويسنده , , Paul A. and Zaytzev، نويسنده , , Andrey V. and Whitwood، نويسنده , , Adrian C.، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2007
  • Pages
    4
  • From page
    5209
  • To page
    5212
  • Abstract
    The diastereoselective pot, atom and step economic (PASE) synthesis of highly functionalized piperidines has been realized. The procedure simply involves mixing methyl acetoacetate, 2 equiv of aldehyde and 2 equiv of aniline together in the presence of InCl3. In most cases the piperidine precipitates out of solution.
  • Keywords
    piperidines , PASE , One-pot , Multi-component
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2007
  • Journal title
    Tetrahedron Letters
  • Record number

    1855699