Title of article :
Efficient reductive acylation of 3-nitroindoles
Author/Authors :
Roy، نويسنده , , Sujata and Roy، نويسنده , , Sudipta and Gribble، نويسنده , , Gordon W.، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2008
Abstract :
3-Nitroindoles are catalytically reduced by hydrogen on palladium/carbon to furnish the relatively unstable aminoindoles, which in the presence of carboxylic acid anhydrides afford good to excellent yields of the corresponding N-acylaminoindoles. 2-Nitroindoles give lower yields of N-acylated 2-aminoindoles.
Keywords :
Acylaminoindoles , Nitroindoles , Hydrogenation , Aminoindoles , Reduction
Journal title :
Tetrahedron Letters
Journal title :
Tetrahedron Letters