• Title of article

    A general method for regioselective Heck arylation of electron-rich N-acyl-N-vinylamine with aryl halides

  • Author/Authors

    Liu، نويسنده , , Zhihua and Xu، نويسنده , , Zheng-Dan and Tang، نويسنده , , Weijun and Xu، نويسنده , , Lijin and Mo، نويسنده , , Jun and Xiao، نويسنده , , Jianliang، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2008
  • Pages
    5
  • From page
    2756
  • To page
    2760
  • Abstract
    A highly efficient protocol for the Pd-catalyzed regioselective Heck arylation of the electron-rich olefin N-acyl-N-vinylamine with aryl halides has been developed. In the presence of hydrogen-bond donor [H2NiPr2][BF4] as an additive, this proceeds smoothly in isopropanol to afford exclusively the branched products in high yields.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2008
  • Journal title
    Tetrahedron Letters
  • Record number

    1859006