A direct route to triazole boronic esters and their application in the synthesis of small molecule arrays
Author/Authors :
Huang، نويسنده , , Jianhui and Macdonald، نويسنده , , Simon J.F. and Cooper، نويسنده , , Anthony W.J. and Fisher، نويسنده , , Gail and Harrity، نويسنده , , Joseph P.A. Harrity، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2009
Pages :
3
From page :
5539
To page :
5541
Abstract :
Alkynylboronates represent useful substrates for the direct synthesis of triazole boronic esters by their thermal cycloaddition with azides. A telescoped cycloaddition–cross-coupling protocol is reported and its employment in the synthesis of a small triazole array is disclosed.
