Title of article
Highly efficient one-pot C-, N- and O-acylation of indolin-2-one analogs
Author/Authors
Jha، نويسنده , , Mukund and Blunt، نويسنده , , Brian، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2009
Pages
4
From page
6044
To page
6047
Abstract
A highly efficient one-pot multiple acylation at chemically non-equivalent sites on indolin-2-one and related motifs using 4-(N,N-dimethylamino)pyridine as a catalyst is described. This procedure gives extremely facile entry to highly desired 3-acyl-2-hydroxy-indole synthons among other derivatives.
Keywords
3-Acetyl-2-hydroxyindole , Multiple acylation , DMAP , acetylation , indole , Indolin-2-one , Indoline-2-thione
Journal title
Tetrahedron Letters
Serial Year
2009
Journal title
Tetrahedron Letters
Record number
1866324
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