• Title of article

    Parallel synthesis enablement of 2-pyridyl-5-cyano-pyrimidine-6-ones—a novel class of HIF-hydroxylase inhibitors

  • Author/Authors

    Chang، نويسنده , , Shang-Poa and Hungerford، نويسنده , , William M. and McDonald، نويسنده , , Wayne S. and Maguire، نويسنده , , Robert J. and Malony، نويسنده , , Kelly Q. and Subramanyam، نويسنده , , Chakrapani، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2010
  • Pages
    3
  • From page
    952
  • To page
    954
  • Abstract
    The synthesis of various substituted 2-pyridyl-5-cyano-pyrimidine-6-ones was accomplished via a three-step protocol. The key aspects of this parallel protocol was the preparation of amidines from nitriles under mild conditions followed by cyclization with ethyl (ethoxymethylene)cyanoacetate.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2010
  • Journal title
    Tetrahedron Letters
  • Record number

    1871074