• Title of article

    Nitrogen ylide-mediated cyclopropanation of lactams and lactones

  • Author/Authors

    Villar، نويسنده , , Irene Suarez del and Gradillas، نويسنده , , Ana and Domيnguez-Romero، نويسنده , , Gema and Pérez-Castells، نويسنده , , Javier، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2010
  • Pages
    4
  • From page
    3095
  • To page
    3098
  • Abstract
    Cyclopropanation of α,β-unsaturated δ-lactams and δ-lactones mediated by nitrogen ylides is described. The process tolerates different alkyl halides and gives efficiently bicyclo[4.1.0]heptanes in a totally stereoselective manner. On the other hand, ε-lactams under our experimental conditions suffer a novel process involving a skeletal reorganization to give a bicyclic[3.3.0] system.
  • Keywords
    Cyclopropanation , Lactones , lactams , Nitrogen ylides , Rearrangements
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2010
  • Journal title
    Tetrahedron Letters
  • Record number

    1872274