Author/Authors :
White، نويسنده , , James R. and Price، نويسنده , , Gareth J. and Schiffers، نويسنده , , Stefanie and Raithby، نويسنده , , Paul R. and Plucinski، نويسنده , , Pawel K. and Frost، نويسنده , , Christopher G.، نويسنده ,
Abstract :
The stable benzylazido-boronate ester 1 is presented as an example of a dual-functional linker that allows the synthetically valuable boronate motif to be clicked onto other molecules under mild conditions. The utility of the azido-boronate motif as a modular building block is demonstrated in the rapid synthesis of drug-like structures employing sequential catalytic azide–alkyne cycloaddition and Suzuki coupling reactions.
