Author/Authors :
Sakya، نويسنده , , Subas M. and Van Den Berg، نويسنده , , Michel and Pouwer، نويسنده , , Kees and Humphrey، نويسنده , , John M. and Helal، نويسنده , , Christopher J. and O’Donnell، نويسنده , , Christopher J.، نويسنده ,
Abstract :
2,3-Azaisoindoline (4) was prepared via reaction of dichloride 11 with 2,4-dimethoxybenzyl amine followed by deprotection with trifluoroacetic acid and triethylsilane. Isolation of the unstable 2,3-azaisoindoline 4 was facilitated by conversion to the bis-HCl salt.