Title of article
Synthesis of 4-aza analog of ramelteon: a novel tricyclic 1,6,7,8-tetrahydro-2H-cyclopenta[d]furo[2,3-b]pyridine derivative as melatonin receptor ligand
Author/Authors
Koike، نويسنده , , Tatsuki and Hoashi، نويسنده , , Yasutaka and Takai، نويسنده , , Takafumi and Uchikawa، نويسنده , , Osamu، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2011
Pages
3
From page
3009
To page
3011
Abstract
The 4-aza analog of ramelteon (−)-1, a novel tricyclic 1,6,7,8-tetrahydro-2H-cyclopenta[d]furo[2,3-b]pyridine derivative, was synthesized via the intramolecular inverse electron demand Diels–Alder reaction followed by fluoride-induced desilylation–cyclization.
Keywords
intramolecular Diels–Alder reaction , 3-b]pyridine , Ramelteon , Desilylation–cyclization
Journal title
Tetrahedron Letters
Serial Year
2011
Journal title
Tetrahedron Letters
Record number
1878451
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