• Title of article

    Synthesis of resorcin[4]arene bearing self-folding substituent

  • Author/Authors

    Enmi، J. نويسنده , , Yoshinori and Kobayashi، نويسنده , , Kazuhiro and Konishi، نويسنده , , Hisatoshi and Morimoto، نويسنده , , Minoru، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2011
  • Pages
    4
  • From page
    3367
  • To page
    3370
  • Abstract
    Thiomethylation of resorcin[4]arene using N,N-diisopropyl-2-aminoethanethiol hydrochloride and formaldehyde [1:4:4 molar ratio] carried out in methanol/acetic acid [1:1 v/v] at 60 °C produced monofunctionalized product 3 in 68% yield. The introduced substituent was intramolecularly self-included into the cavity. This self-inclusion reduced the reactivity of the aromatic rings and inhibited further functionalization.
  • Keywords
    Thiomethylation , Self-inclusion , Monofunctionalization
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2011
  • Journal title
    Tetrahedron Letters
  • Record number

    1878617