• Title of article

    Cernumidine and isocernumidine, new type of cyclic guanidine alkaloids from Solanum cernuum

  • Author/Authors

    Lopes، نويسنده , , Luciane C. and Roman، نويسنده , , Bianca and Medeiros، نويسنده , , Maria A. and Mukhopadhyay، نويسنده , , Abhik and Utrilla، نويسنده , , Pilar and Gلlvez، نويسنده , , Julio and Mauriٌo، نويسنده , , Sofيa Garcيa and Moltiva، نويسنده , , Virginia and Lourenço، نويسنده , , Ana and Feliciano، نويسنده , , Arturo San Feliciano، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2011
  • Pages
    4
  • From page
    6392
  • To page
    6395
  • Abstract
    Cernumidine and isocernumidine were identified in the ethanol extract of the leaves of Solanum cernuum Vell. together with four known phenolic compounds. The alkaloids have a natural (2-aminopyrrolidin-1-yl)carboxamidine alkaloidal base acylated with isoferulic (3-hydroxy-4-methoxycinnamic) acid with Z and E configurations, respectively. The structures were elucidated on the basis of 1D- and 2D-NMR data and the structure of cernumidine was confirmed by X-ray analysis. Cernumidine displayed inhibition of interleukin-8 production by HT-29 colon carcinoma cells. This fact could orient further research in gastric cancer prevention and treatment.
  • Keywords
    Alkaloids , Cernumidines , Solanum cernnum Vell. , interleukin-8
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2011
  • Journal title
    Tetrahedron Letters
  • Record number

    1879613