Title of article
Microwave-assisted aza-Prins reaction. Part 1: facile preparation of natural-like 3-azabicyclo[3.3.1]non-6-enes
Author/Authors
Parchinsky، نويسنده , , Vladislav and Shumsky، نويسنده , , Alexei and Krasavin، نويسنده , , Mikhail، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2011
Pages
4
From page
7157
To page
7160
Abstract
A facile and operationally simple route to diastereomerically pure, natural-like 3-azabicyclo[3.3.1]non-6-enes via microwave-assisted, BF3·OEt2-promoted aza-Prins reaction has been developed. Complexity-generating transformations based on these products involving reactive functionalities introduced during the aza-Prins step have been developed.
Keywords
diastereoselective synthesis , Bicyclic piperidines , lycopodium alkaloids , Complexity-generating synthesis , Microwave-assisted organic synthesis , aza-Prins reaction
Journal title
Tetrahedron Letters
Serial Year
2011
Journal title
Tetrahedron Letters
Record number
1879802
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