• Title of article

    Efficient synthesis of kaempferol 3,7-O-bisglycosides via successive glycosylation with glycosyl ortho-alkynylbenzoates and trifluoroacetimidates

  • Author/Authors

    Yang، نويسنده , , Weizhun and Sun، نويسنده , , Jiansong and Yang، نويسنده , , Zhongyi and Han، نويسنده , , Wei and Zhang، نويسنده , , Wei-Dong and Yu، نويسنده , , Biao، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2012
  • Pages
    4
  • From page
    2773
  • To page
    2776
  • Abstract
    Selective glycosylation of the 3-OH of 5,4′-di-O-acetyl-kaempferol was achieved with glycosyl ortho-alkynylbenzoates as donors under the catalysis of Ph3PAuNTf2, and subsequent glycosylation of the remaining 7-OH with glycosyl trifluoroacetimidates under the catalysis of BF3·OEt2, after global deprotection, afforded the kaempferol 3,7-O-bisglycosides conveniently.
  • Keywords
    kaempferol , Selective glycosylation , Glycosyl ortho-alkynylbenzoate , glycosyl trifluoroacetimidate
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2012
  • Journal title
    Tetrahedron Letters
  • Record number

    1880838