• Title of article

    Chiral dihydrobenzofuran-based diphosphine (BICMAP): optical resolution and application to rhodium(I)-catalyzed asymmetric 1,4-addition of aryl- and alkenylboronic acids to cyclic enones

  • Author/Authors

    Mino، نويسنده , , Takashi and Hashimoto، نويسنده , , Masatoshi and Uehara، نويسنده , , Katsunori and Naruse، نويسنده , , Yoshiaki and Kobayashi، نويسنده , , Shohei and Sakamoto، نويسنده , , Masami and Fujita، نويسنده , , Tsutomu، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2012
  • Pages
    3
  • From page
    4562
  • To page
    4564
  • Abstract
    Chiral dihydrobenzofuran-based diphosphine ligand (BICMAP) 1 was used as a ligand for the rhodium(I)-catalyzed asymmetric 1,4-addition of arylboronic acids to cyclic enones up to 99% ee. We also found that the BICMAP-rhodium system was an efficient catalyst for the 1,4-addition of alkenylboronic acids to 2-cyclohexenone in good enantioselectivities.
  • Keywords
    Asymmetric reaction , 1 , 4-addition , Rhodium catalyst , Diphosphine
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2012
  • Journal title
    Tetrahedron Letters
  • Record number

    1881609