Title of article
Efficient syntheses of 2-fluoroalkylbenzimidazoles and -benzothiazoles
Author/Authors
René، نويسنده , , Olivier and Souverneva، نويسنده , , Alexandra and Magnuson، نويسنده , , Steven R. and Fauber، نويسنده , , Benjamin P.، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2013
Pages
4
From page
201
To page
204
Abstract
We report an efficient one-step route to 2-fluoroalkylbenzimidazoles and -benzothiazoles via the condensation of fluorinated carboxylic acids and aromatic diamines or aminothiophenols. Additionally, we describe the syntheses of fluoroalkyl-azabenzimidazoles, -purines, and -imidazolopyrazines. This method is high-yielding with broad scope and is operationally simple with potential application to parallel synthesis.
Keywords
Fluoroalkylheterocycles , Purine , Azabenzimidazole , benzothiazole , Benzimidazole
Journal title
Tetrahedron Letters
Serial Year
2013
Journal title
Tetrahedron Letters
Record number
1883345
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