• Title of article

    Efficient synthesis of bicyclo[3.2.1]octane-2,4-diones and their incorporation into potent HPPD inhibitors

  • Author/Authors

    Baalouch، نويسنده , , Myriam and De Mesmaeker، نويسنده , , Alain and Beaudegnies، نويسنده , , Renaud، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2013
  • Pages
    5
  • From page
    557
  • To page
    561
  • Abstract
    Herein we report a very efficient access to a variety of bicyclic 1,3-diones as key intermediates to be incorporated into very potent HPPD inhibitors. In particular, we have developed a one-pot process for the synthesis of the bicyclo[3.2.1]octane-2,4-dione, the parent dione of Bicyclopyrone.
  • Keywords
    HPPD inhibitors , Diels–Alder cycloadditions , Cyclopropene , Bicyclic diones
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2013
  • Journal title
    Tetrahedron Letters
  • Record number

    1883560