Title of article
Novel synthesis of 4,4-difluoropyrido[4,3-b]indoles via intramolecular Heck reaction
Author/Authors
Madaiah، نويسنده , , M. S. Prashanth، نويسنده , , M.K. and Revanasiddappa، نويسنده , , H.D.، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2013
Pages
4
From page
1424
To page
1427
Abstract
Various difluoropyridoindoles were synthesized via a palladium-catalyzed intramolecular Heck reaction as a key step. Thus, ortho-bromoanilines and difluoropiperidinone were treated with (PPh3)2PdCl2 and base in pyridine to give the regioselective cyclized heterocycles in modest to satisfactory yields.
Keywords
Difluoropyridoindole , PALLADIUM , pyridine , Heck reaction , regioselective
Journal title
Tetrahedron Letters
Serial Year
2013
Journal title
Tetrahedron Letters
Record number
1883950
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