Title of article
Simple approach to the synthesis of 3-fluoro pyrazolo[1,5-a]pyrimidine analogues
Author/Authors
Bel Abed، نويسنده , , Hassen and Mammoliti، نويسنده , , Oscar and Van Lommen، نويسنده , , Guy and Herdewijn، نويسنده , , Piet، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2013
Pages
3
From page
2612
To page
2614
Abstract
A simple method for the synthesis of novel 3-fluoro pyrazolo[1,5-a]pyrimidine analogues has been developed starting from fluoro acetonitrile and benzoyl chloride. The desired compounds are synthesized from a 3-amino-4-fluoro pyrazole intermediate. The versatility of the approach was demonstrated by the synthesis of a small library of pyrazolo[1,5-a]pyrimidine.
Keywords
5-a]pyrimidine , heterocycle , cyclization , Pyrazole
Journal title
Tetrahedron Letters
Serial Year
2013
Journal title
Tetrahedron Letters
Record number
1884451
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