Title of article :
Synthesis of oxygenated 2-methylindolines
Author/Authors :
Chang، نويسنده , , Meng-Yang and Chen، نويسنده , , Yi-Chia and Chan، نويسنده , , Chieh-Kai، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2014
Abstract :
A palladium-mediated high-yielding synthesis of oxygenated 2-methylindolines 4 from 2-allylnitrobenzene 1 and hydrazine is developed. The one-pot route combines the reduction of 2-allylnitrobenzene 1 and the sequential intramolecular hydroamination. The protocol provides a novel alternative for the synthesis of substituted 2-methylindoline 4.
Keywords :
Hydroamination , 2-Methylindolines , 2-Allylnitrobenzenes
Journal title :
Tetrahedron Letters
Journal title :
Tetrahedron Letters