• Title of article

    Aryl methyl sulfides via SNAr using DMSO as the source of the thiomethyl moiety

  • Author/Authors

    Jones-Mensah، نويسنده , , Ebenezer and Magolan، نويسنده , , Jakob، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2014
  • Pages
    4
  • From page
    5323
  • To page
    5326
  • Abstract
    A unique synthesis of aryl methyl sulfides is reported proceeding via reduction of dimethylsulfoxide to dimethylsulfide at elevated temperature in the presence of Hunig’s base followed by nucleophilic aromatic substitution and demethylation. Activated aryl fluorides, chlorides, and nitrobenzenes are suitable substrates with 13 examples provided. Dimethylsulfoxide serves as a simple and inexpensive formal source of the thiomethyl moiety.
  • Keywords
    Dimethylsulfoxide , nucleophilic aromatic substitution , Methyl sulfides , Thiomethyl , Hunig’s base
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2014
  • Journal title
    Tetrahedron Letters
  • Record number

    1890720