Title of article :
Synthesis of dihydropyrazolo[4,3-c]azepines via iodine-mediated intramolecular hydrative cyclization
Author/Authors :
Batchu، نويسنده , , Harikrishna and Batra، نويسنده , , Sanjay، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2014
Abstract :
A straightforward approach to substituted dihydropyrazolo[4,3-c]azepines via I2-mediated intramolecular hydration in pyrazole-based allylamines prepared from Morita–Baylis–Hillman adducts of 4-iodopyrazolealdehyes is described.
Keywords :
Morita–Baylis–Hillman , Hydrative cyclization , nitrogen heterocycle , iodine , allylamine
Journal title :
Tetrahedron Letters
Journal title :
Tetrahedron Letters