• Title of article

    Catalyst free synthesis of indole derivatives via multicomponent reaction of aniline under solvent-free conditions

  • Author/Authors

    Ghasemian Dazmiri, Mahboubeh Department of Chemistry - Faculty of Sciences - Babolsar University, Mazandaran , Ghasemi, Narges National Petrochemical Company (NPC) - petrochemical Research and Technology Company - Arak Center, Arak , Noushin, Annataj Department of Chemistry - Islamic Azad University Gorgan Branch, Gorgan

  • Pages
    5
  • From page
    3031
  • To page
    3035
  • Abstract
    Protonation of the highly reactive 1:1 intermediates produced in the reaction between alkyl(aryl) isocyanides and dibenzoylacetylene by isatin, leads to vinylnitrilium cations, which undergo carbon-centered Michael type addition with the conjugate base of the NH-acid to produce highly functionalized indole-2,3-diones.
  • Keywords
    Activated acetylenic compounds , Aniline , Alkyl(aryl) isocyanides
  • Journal title
    Iranian Journal of Organic Chemistry
  • Serial Year
    2021
  • Record number

    2703331