• Title of article

    Nitrogen transfer in E. coli glucosamine-6P synthase. Investigations using substrate and bisubstrate analogs

  • Author/Authors

    Marie-Ange Badet-Denisot، نويسنده , , Caroline Leriche، نويسنده , , Frédéric Massière، نويسنده , , Bernard Badet، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1995
  • Pages
    6
  • From page
    815
  • To page
    820
  • Abstract
    The compound 2-amino-2-deoxyglucitol-6P competitively inhibits E. coli glucosamine-6P synthase with respect to fructose-6P whereas glutamate γ-semialdehyde is a competitive inhibitor with respect to glutamine. These compounds, which exhibit good inhibitory properties (Km/Ki= 16 and 1000 respectively), were used in the synthesis of multisubstrate analogs.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1995
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    787421