Title of article
Synthesis and evaluation of 2-aryl-4H-3,1-benzoxazin-4-ones as C1r serine protease inhibitors
Author/Authors
John L. Gilmore، نويسنده , , Sheryl J. Hays، نويسنده , , Bradley W. Caprathe، نويسنده , , Chitase Lee، نويسنده , , Mark R. Emmerling، نويسنده , , Walter Michael Halbmayer، نويسنده , , Juan C. Jaen، نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 1996
Pages
4
From page
679
To page
682
Abstract
A series of 2-aryl-4H-3,1-benzoxazin-4-ones have been synthesized and tested for inhibitory activity against C1r serine protease. Compounds were found that were equipotent and more selective than the reference compound FUT-175.
Journal title
Bioorganic & Medicinal Chemistry Letters
Serial Year
1996
Journal title
Bioorganic & Medicinal Chemistry Letters
Record number
787980
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