Title of article :
BMS-187257, a potent, selective, and novel heterocyclic β3 adrenergic receptor agonist
Author/Authors :
Liesl G. Fisher، نويسنده , , Philip M. Sher، نويسنده , , Stephen Skwish، نويسنده , , Inge M. Michel، نويسنده , , Steven M. Seiler، نويسنده , , Kenneth E. J. Dickinson، نويسنده ,
Issue Information :
روزنامه با شماره پیاپی سال 1996
Abstract :
Novel heterocyclic β3 adrenergic receptor agonists2 were prepared and evaluated for their ability to bind to human β1, β2, and β3 adrenergic receptors. Stimulatory effects on the β3 adrenergic receptor were also measured. BMS-187257 (4b) was found to be a potent and selective β3 agonist.
Journal title :
Bioorganic & Medicinal Chemistry Letters
Journal title :
Bioorganic & Medicinal Chemistry Letters
