Title of article :
Double activation preparation of an acridinyl-isoxazolyl-lexitropsin
Author/Authors :
Peiwen Zhou، نويسنده , , Michael D. Mosher، نويسنده , , Wendy D. Taylor، نويسنده , , Gregory A. Crawford، نويسنده , , N. R. Natale، نويسنده ,
Issue Information :
روزنامه با شماره پیاپی سال 1997
Abstract :
The coupling of a sterically hindered acridinyl isoxazole ester directly to the amine group of a lexitropsin is significantly improved by double activation, using trimethylaluminum to activate the amine portion and samarium (III) chloride to enhance the carboxylate reactivity.
Journal title :
Bioorganic & Medicinal Chemistry Letters
Journal title :
Bioorganic & Medicinal Chemistry Letters