Title of article
Targeting DNA topoisomerase II with podophyllotoxin aza-analogue
Author/Authors
Akira Iida، نويسنده , , Masahiro Kano، نويسنده , , Yoshihiro Kubota، نويسنده , , Kenji Koga and Harutoshi Takeo، نويسنده , , Kiyoshi Tomioka، نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 1997
Pages
2
From page
2565
To page
2566
Abstract
Oxidation of a cytotoxic podophyllotoxin aza-analogue 2 into the quinone 3succeeded in acquiring DNA topoisomerase II inhibitory activity at a concentration of 25 μM due to stabilization of the cleavable complex.
Journal title
Bioorganic & Medicinal Chemistry Letters
Serial Year
1997
Journal title
Bioorganic & Medicinal Chemistry Letters
Record number
789003
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