Author/Authors :
Kazuo Kubo، نويسنده , , Toshiyuki Shimizu، نويسنده , , Shin-ichi Ohyama، نويسنده , , Hideko Murooka، نويسنده , , Tsuyoshi Nishitoba، نويسنده , , Shinichiro Kato، نويسنده , , Yoshiko Kobayashi، نويسنده , , Mikio Yagi، نويسنده , , Toshiyuki Isoe، نويسنده , , Kazuhide Nakamura، نويسنده , , Tatsushi Osawa، نويسنده , , Toshio Izawa، نويسنده ,
Abstract :
A novel series of 4-phenoxyquinolines, some of which showed potent and highly selective inhibitory activities for PDGF receptor autophosphorylation, was discovered. Interestingly, their structures were very similar to those of the selective inhibitors for EGF receptor autophosphorylation.