• Title of article

    Design and synthesis of a water-soluble taxol analogue : Taxol-sialyl conjugate

  • Author/Authors

    Takashi Takahashi، نويسنده , , Hirokazu Tsukamoto، نويسنده , , Haruo Yamada، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1998
  • Pages
    4
  • From page
    113
  • To page
    116
  • Abstract
    Glycosidation, using the methylthio derivative of N-acetylneuraminic acid 3, of linker alcohol 4 in DME with “long-range participation” produced the α-glycosyl linkage with high stereoselectivity. The α-linked sialic acid 2 was introduced in taxol without protection of the alcohol functionality in sialic acid.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1998
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    789189