• Title of article

    Synthesis and antibacterial activity of [6,5,5] and [6,6,5] tricyclic fused oxazolidinones

  • Author/Authors

    D. Mark Gleave، نويسنده , , Steven J. Brickner، نويسنده , , Peter R. Manninen، نويسنده , , Debra A. Allwine، نويسنده , , Kristine D. Lovasz، نويسنده , , Douglas C. Rohrer، نويسنده , , John A. Tucker، نويسنده , , Gary E. Zurenko، نويسنده , , Charles W. Ford، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1998
  • Pages
    6
  • From page
    1231
  • To page
    1236
  • Abstract
    A series of conformationally restricted, [6,5,5] and [6,6,5] tricyclic fused oxazolidinones were synthesized and tested for antibacterial activity. Several compounds in the trans-[6,5,5] series demonstrated potent in vitro and in vivo activity. This work provides valuable information regarding the preferred conformational orientation of the oxazolidinones at the binding site.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1998
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    789409