• Title of article

    Synthesis and evaluation of artificial taxoids with antitumor and multi-drug resistance reversing activities

  • Author/Authors

    Koichiro Morihira، نويسنده , , Toshiyuki Nishimori، نويسنده , , Hiroyuki Kusama، نويسنده , , Yoshiaki Horiguchi، نويسنده , , Isao Kuwajima، نويسنده , , Takashi Tsuruo، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1998
  • Pages
    6
  • From page
    2977
  • To page
    2982
  • Abstract
    Artificial taxoids were synthesized and subjected to evaluation of their ability of multi-drug resistance reversing and antitumor activities. While the taxoid 4 could not increase cellular accumulation of vincristine in multi-drug resistant tumor cells, the C4-hydroxy analog 15 showed significant effect. However, these compounds showed weak activities on growth inhibition of cancer cells.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1998
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    789742