• Title of article

    Syntheses of novel antitumor dihydroxanthone derivatives with inhibitory activity against DNA topoisomerase II

  • Author/Authors

    Seiichi Sato، نويسنده , , Yasuyo Suga، نويسنده , , Toshihiko Yoshimura، نويسنده , , Ryusuke Nakagawa، نويسنده , , Takashi Tsuji، نويسنده , , Ken Umemura، نويسنده , , Toshiwo Andoh، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1999
  • Pages
    4
  • From page
    2653
  • To page
    2656
  • Abstract
    A series of methoxycarbonyl group modified nidulalin A analogs were synthesized to improve stability against esterases. The amide derivatives showed cytotoxic activity along with inhibitory activity against DNA topoisomerase II. Among the analogs, amide 9a exhibited antitumor activity in Colon 26 murine tumor model.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1999
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    790400