• Title of article

    4-Thiazolidinones: novel inhibitors of the bacterial enzyme murB

  • Author/Authors

    Charles J. Andres، نويسنده , , Joanne J. Bronson، نويسنده , , Stanley V. DʹAndrea، نويسنده , , Milind S. Deshpande، نويسنده , , Paul J. Falk، نويسنده , , Katharine A. Grant-Young، نويسنده , , William E. Harte، نويسنده , , Hsu-Tso Ho، نويسنده , , Peter F. Misco، نويسنده , , James G. Robertson، نويسنده , , David Stock، نويسنده , , Yaxiong Sun، نويسنده , , Ann W. Walsh، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2000
  • Pages
    3
  • From page
    715
  • To page
    717
  • Abstract
    4-Thiazolidinones were synthesized and evaluated for their ability to inhibit the bacterial enzyme MurB. Selected 4-thiazolidinones displayed activity against the enzyme in vitro. This activity, coupled with the design principles of the thiazolidinones, supports the postulate that 4-thiazolidinones may be recognized as diphosphate mimics by a biological selector.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2000
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    790722