• Title of article

    The design and synthesis of the high efficacy, non-peptide CCK1 receptor agonist PD 170292

  • Author/Authors

    N. Bernad، نويسنده , , B. G. M. Burgaud، نويسنده , , D. C. Horwell، نويسنده , , R. A. Lewthwaite، نويسنده , , J. Martinez، نويسنده , , M. C. Pritchard، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2000
  • Pages
    4
  • From page
    1245
  • To page
    1248
  • Abstract
    The design, synthesis and biological actions of a novel, non-peptide CCK1 receptor agonist (PD 170292) which exhibits a similar pharmacological profile to the CCK analogue JMV180 is reported. PD 170292 was designed based on a consideration of the structures of a peptide based CCK1 receptor selective agonist and a peptoid CCK2 receptor selective antagonist.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2000
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    790843