• Title of article

    Discovery of a potent, non-triketone type inhibitor of 4-hydroxyphenylpyruvate dioxygenase

  • Author/Authors

    Shean-woei Lin، نويسنده , , Yun-Loung Lin، نويسنده , , Tzu-Ching Lin، نويسنده , , Ding-Yah Yang، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2000
  • Pages
    2
  • From page
    1297
  • To page
    1298
  • Abstract
    3-Cyclopropanecarbonyloxy-2-cyclohexen-1-one has been found to be a new, potent, low molecular weight non-triketone type inhibitor of 4-hydroxyphenylpyruvate dioxygenase with IC50 value of 30 nM. Preliminary studies suggest that the two carbonyl groups present in the compound are crucial for the inhibition activity.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2000
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    790856