Title of article
2,4,5-Trisubstituted imidazoles: novel nontoxic modulators of P-glycoprotein mediated multidrug resistance. Part 1[]
Author/Authors
Sepehr Sarshar، نويسنده , , Chengzhi Zhang، نويسنده , , Edmund J. Moran، نويسنده , , Sonja Krane، نويسنده , , Jennifer C. Rodarte، نويسنده , , Khalid D. Benbatoul، نويسنده , , Ross Dixon، نويسنده , , Adnan M. M. Mjalli، نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 2000
Pages
3
From page
2599
To page
2601
Abstract
N-4,5-Di-(4-dialkylamino)phenyl imidazoles (A) are potent modulators of P-glycoprotein mediated multidrug resistance. This manuscript describes the discovery and lead optimization of this novel class of inhibitors.
Journal title
Bioorganic & Medicinal Chemistry Letters
Serial Year
2000
Journal title
Bioorganic & Medicinal Chemistry Letters
Record number
791162
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