• Title of article

    Importance of the C28–C38 hydrophobic domain of okadaic acid for potent inhibition of protein serine-threonine phosphatases 1 and 2A

  • Author/Authors

    Valerie A. Frydrychowski، نويسنده , , Rebecca A. Urbanek، نويسنده , , Amy B. Dounay، نويسنده , , Craig J. Forsyth، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2001
  • Pages
    3
  • From page
    647
  • To page
    649
  • Abstract
    Okadaic acid is a potent inhibitor of select serine/threonine protein phosphatases. The importance of the C28–C38 hydrophobic domain of okadaic acid for inhibition of PP1 and PP2A was investigated. The hydrophobic domain is required but not sufficient for potent inhibition, and it also contributes to differential inhibition between PP1 and PP2A.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2001
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    791243