• Title of article

    Novel synthesis and RNA-Binding properties of aminoglycoside dimers conjugated via a naphthalene diimide-based intercalator

  • Author/Authors

    Jeffrey B. -H. Tok، نويسنده , , Jason Fenker، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2001
  • Pages
    5
  • From page
    2987
  • To page
    2991
  • Abstract
    The synthesis and RNA-binding properties of naphthalene-based diimide conjugated bis-aminoglycoside antibiotics are reported. Compared to the monomeric aminoglycoside, the conjugated ligands were observed to attain up to 35-fold enhancement in binding affinity towards a novel RNA construct that contained two 16S rRNA A-sites.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2001
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    791776