Title of article
New Generation Dopaminergic Agents. Part 8: Heterocyclic Bioisosteres that Exploit the 7-OH-2-(aminomethyl)chroman D2 Template
Author/Authors
Richard E. Mewshaw، نويسنده , , Rulin Zhao، نويسنده , , Xiaojie Shi، نويسنده , , Karen Marquis، نويسنده , , Julie A. Brennan، نويسنده , , Hossein Mazandarani، نويسنده , , Joseph Coupet، نويسنده , , Terrance H. Andree، نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 2002
Pages
4
From page
271
To page
274
Abstract
Based on the 7-OH-2-(aminomethyl)chroman dopamine D2 template (2) is described the preparation and resolution of two bioisosteric analogues. The benzimidazol-2-one derivative (6) had similar affinity to the known indolone derivative (4).
Journal title
Bioorganic & Medicinal Chemistry Letters
Serial Year
2002
Journal title
Bioorganic & Medicinal Chemistry Letters
Record number
791951
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