Author/Authors :
John A. Lowe III، نويسنده , , Susan E. Drozda، نويسنده , , Katherine Fisher، نويسنده , , Christine Strick، نويسنده , , Lorraine Lebel، نويسنده , , Christopher Schmidt، نويسنده , , Donna Hiller، نويسنده , , Kathleen S. Zandi، نويسنده ,
Abstract :
The synthesis of NPTS, 6, a potent inhibitor of the type 1 glycine transporter (GlyT1) is described, as well as preparation of 6 in optically active and tritiated form for use as a radioligand for affinity displacement assay of GlyT1.