• Title of article

    Chemical synthesis and cytotoxicity of dihydroxylated cyclopentenone analogues of neocarzinostatin chromophore

  • Author/Authors

    Michael D. Urbaniak، نويسنده , , Lisa M. Frost، نويسنده , , John P. Bingham، نويسنده , , Lloyd R. Kelland، نويسنده , , John A. Hartley، نويسنده , , Derek N. Woolfson، نويسنده , , Stephen Caddick، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2003
  • Pages
    3
  • From page
    2025
  • To page
    2027
  • Abstract
    Compounds containing the naphthoate moiety of Neocarzinostatin chromophore or 2-hydroxynaphthoate have been synthesized and evaluated for cytotoxic activity against a leukemia cell line and a small panel of human-tumor cell lines. Those compounds containing a cyclopentenone moiety were active, with the carbonyl group being essential for biological activity.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2003
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    793289