• Title of article

    Glycidol-carbohydrate hybrids: a new family of DNA alkylating agents

  • Author/Authors

    Kazunobu Toshima، نويسنده , , Yukiko Okuno، نويسنده , , Shuichi Matsumura، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2003
  • Pages
    3
  • From page
    3281
  • To page
    3283
  • Abstract
    Novel and chiral glycidol–carbohydrate hybrids possessing an epoxy group as a DNA alkylating moiety were designed and synthesized. These artificial hybrids selectively alkylated DNA at the N-7 sites of the guanines and cleaved DNA without any additives. The binding ability of the glycidol was significantly enhanced by the attachment of the carbohydrate.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2003
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    793553