Title of article
Biological evaluation of substituted quinolines
Author/Authors
Xavier Franck، نويسنده , , Alain Fournet، نويسنده , , Eric Prina، نويسنده , , Renaud Mahieux، نويسنده , , Reynald Hocquemiller، نويسنده , , Bruno Figadere، نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 2004
Pages
4
From page
3635
To page
3638
Abstract
Several quinolines were synthesized and evaluated in vitro against several parasites (Trypanosoma brucei, T. cruzi, Leishmania infantum, L. amazonensis, Plasmodium falciparum). Then, they were evaluated in vitro (at 10 μM), against HTLV-1 transformed cells. A few of them displayed interesting activities, comparable to the reference drugs.
Keywords
Protozoa , HTLV-1 , Leishmaniases , Trypanozomiases.* Corresponding author. Tel.: +33-01-46-83-55-92 , fax:+33-01-46-83-53-99 , e-mail: bruno.figadere@cep.u-psud.fr
Journal title
Bioorganic & Medicinal Chemistry Letters
Serial Year
2004
Journal title
Bioorganic & Medicinal Chemistry Letters
Record number
794651
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