• Title of article

    Efficient cleavage of RNA, enhanced cellular uptake, and controlled intracellular localization of conjugate DNAzymes

  • Author/Authors

    Takanori Kubo، نويسنده , , Kengo Takamori، نويسنده , , Kenichi Kanno، نويسنده , , Bakalova Rumiana، نويسنده , , Hideki Ohba، نويسنده , , Miho Matsukisono، نويسنده , , Yasuo Akebiyama، نويسنده , , Masayuki Fujii، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2005
  • Pages
    4
  • From page
    167
  • To page
    170
  • Abstract
    Conjugate DNAzymes with polyamines and peptides were successfully prepared by solid phase fragment condensation (SPFC) and showed up to 4.2 times higher catalytic efficiency (kcat/Km) and enhanced tolerance against DNase 1digestion. To be pointed out, intracellular localization of DNAzymes could be controlled by conjugated with naturally occurring signal peptides responsible for nuclear cytoplasmic transport of proteins.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2005
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    795172