Title of article
Synthesis of cyclic peptidosulfonamides as scaffolds for MC4 pharmacophoric groups
Author/Authors
Bas Wels، نويسنده , , John A.W. Kruijtzer، نويسنده , , Keith M. Garner، نويسنده , , Roger A.H. Adan، نويسنده , , Rob M.J. Liskamp، نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 2005
Pages
4
From page
287
To page
290
Abstract
The synthesis of potential β-turn mimetics based on cyclic sulfonamide peptoid/peptoid hybrids is described. These are readily synthesized using a solid phase protocol followed by cyclization in solution, and their suitability to combinatorial approaches is illustrated by the synthesis of a small but diversely functionalized library.
Keywords
Peptoid , MC4-agonists , Cyclic peptide , solid phase synthesis , Peptidosulfonamide , Peptidomimetic
Journal title
Bioorganic & Medicinal Chemistry Letters
Serial Year
2005
Journal title
Bioorganic & Medicinal Chemistry Letters
Record number
795194
Link To Document