Title of article
3H-Quinazolin-4-ones as a new calcilytic template for the potential treatment of osteoporosis
Author/Authors
Irina Shcherbakova، نويسنده , , Manuel F. Balandrin، نويسنده , , John Fox، نويسنده , , Anjan Ghatak، نويسنده , , William L. Heaton، نويسنده , , Rebecca L. Conklin، نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 2005
Pages
4
From page
1557
To page
1560
Abstract
Structure–activity relationship studies, focused on identification of the active pharmacophore fragments in a single high-throughput screening calcilytic hit, resulted in the discovery of potent calcium receptor antagonists, substituted 3H-quinazolin-4-ones.
Keywords
3H-Quinazolin-4-ones , osteoporosis , Calcilytics , Calcium receptor antagonists
Journal title
Bioorganic & Medicinal Chemistry Letters
Serial Year
2005
Journal title
Bioorganic & Medicinal Chemistry Letters
Record number
795434
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